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Open Access Articles- Top Results for Cinolazepam

Cinolazepam

Not to be confused with clonazepam or camazepam.
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Cinolazepam
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Systematic (IUPAC) name
(RS)-3-[9-Chloro-6-(2-fluorophenyl)-4-hydroxy-3-oxo-2,5-diazabicyclo[5.4.0]undeca-5,8,10,12-tetraen-2-yl]propanenitrile
Clinical data
AHFS/Drugs.com International Drug Names
  •  ?
Oral
Pharmacokinetic data
Bioavailability 90-100%
Metabolism Hepatic
Half-life 9 h[1]
Excretion Renal
Identifiers
75696-02-5 7pxY
N05CD13
PubChem CID 3033621
DrugBank DB01594 7pxY
ChemSpider 2298251 7pxY
UNII 68P0556B0U 7pxY
KEGG D07328 7pxY
ChEBI CHEBI:59514 7pxY
ChEMBL CHEMBL2104926 7pxN
Chemical data
Formula C18H13ClFN3O2
357.8
 14pxN (what is this?)  (verify)

Cinolazepam[2] (marketed under the brand name Gerodorm)[3] is a drug which is a benzodiazepine derivative. It possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. Due to its strong sedative properties, it is primarily used as an hypnotic.

Cinolazepam is not approved for sale in the United States or Canada.

See also

References

  1. ^ Saletu, B.; G. Kindshofer; P. Anderer; J. Grunberger (1987). "Short-term sleep laboratory studies with cinolazepam in situational insomnia induced by traffic noise.". International Journal of Clinical Pharmacology Research 7 (5): 407–18. PMID 2889679. 
  2. ^ US Patent 4388313 Novel 3-hydroxy-1,4-benzodiazepine-2-ones and process for the preparation thereof
  3. ^ Lannacher Romania (1999). "Gerodorm". Produse Gerot inregistrate in Romania (in Romanian). Archived from the original on 11 October 2006. Retrieved 17 August 2006. 

External links


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